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I-Doxofylline (CAS# 69975-86-6)

Isakhiwo Samakhemikhali:

I-Molecular Formula I-C11H14N4O4
I-Molar Mass 266.25
Ukuminyana 1.2896 (isilinganiso esinzima)
I-Melting Point 144-146°C
I-Boling Point 409.46°C (isilinganiso esinzima)
I-Flash Point 259.3°C
Ukuncibilika kwamanzi Encibilikayo
Ukuncibilika Incibilika emanzini, i-acetone, i-ethyl acetate, i-benzene, i-chloroform, i-dioxane, i-methanol eshisayo noma i-ethanol eshisayo, cishe ayincibiliki ku-ether noma ku-petroleum ether.
I-Vapor Presure 2.49E-10mmHg ku-25°C
Ukubukeka I-Crystallization
Umbala Okumhlophe kuya kokumhlophe
I-Merck 14,3438
pKa 0.42±0.70(Okubikezelwe)
Isimo Sesitoreji ngaphansi kwegesi ye-inert (nitrogen noma i-Argon) ku-2-8°C
I-Refractive Index 1.6000 (isilinganiso)
I-MDL I-MFCD00865218

Imininingwane Yomkhiqizo

Omaka bomkhiqizo

Ubungozi Nokuphepha

Izimpawu Eziyingozi Xi - Irritant
Amakhodi Engozi 36/37/38 - Ukucasula amehlo, uhlelo lokuphefumula kanye nesikhumba.
Incazelo Yokuphepha S26 – Uma uthintana namehlo, geza ngokushesha ngamanzi amaningi futhi ufune iseluleko sezokwelapha.
I-S36/37 – Gqoka izingubo zokuzivikela ezifanele namagilavu.
I-RTECS XH5135000
Ikhodi ye-HS 29399990
Ubuthi I-LD50 kumagundane (mg/kg): 841 ngomlomo; 215.6 iv; kumagundane: 1022.4 ngomlomo, 445 ip (Franzone)

 

I-Doxofylline (CAS# 69975-86-6) Yethula

Sethula i-Doxofylline (CAS# 69975-86-6) - i-bronchodilator eguqulayo eklanyelwe ukuthuthukisa impilo yokuphefumula kanye nokwenza ngcono izinga lempilo yabantu abaphethwe yizimo zokuphefumula ezingapheli. Njengelungu lesigaba semithi ye-xanthine, i-Doxofylline inikeza indlela yokusebenza eyingqayizivele eyenza ihluke kuma-bronchodilators endabuko, okuyenza ibe isengezo esibalulekile ku-arsenal yokwelapha yokuphathwa kwesifuba somoya kanye nesifo esingamahlalakhona sokuvimbela i-pulmonary (COPD).

I-Doxofylline isebenza ngokuphumuza imisipha ebushelelezi yemigudu yomoya, okuholela ekugelezeni komoya okuthuthukisiwe kanye nokuncipha kokucindezeleka kokuphefumula. Isenzo sawo esimbaxambili asigcini nje ngokunweba imigudu ye-bronchial kodwa futhi sinezinto ezilwa nokuvuvukala, ukubhekana nokuvuvukala okucashile okuvame ukwandisa izimo zokuphefumula. Lokhu kwenza i-Doxofylline ibe ukukhetha okusebenzayo ezigulini ezifuna ukukhululeka ekuhefuleni, ukuphelelwa umoya, nezinye izimpawu ezihlobene nesifo somoya kanye ne-COPD.

Esinye sezici ezivelele ze-Doxofylline iphrofayili yayo yokuphepha evumayo. Ngokungafani namanye ama-bronchodilator, mancane amathuba okuthi abangele imiphumela engemihle njenge-tachycardia noma ukuphazamiseka kwamathumbu, okuyenza ifanelekele ukusetshenziswa isikhathi eside. Ukwengeza, i-Doxofylline itholakala ngezindlela ezihlukahlukene, okuhlanganisa amaphilisi nama-inhaler, ehlinzeka ngokuguquguquka kanye lula ezigulini ekulawuleni isimo sazo.

Ngokusebenza kwayo okuqinisekisiwe nokuphepha, i-Doxofylline isiba yinketho ekhethwayo ngokushesha phakathi kochwepheshe bezokunakekelwa kwempilo. Inika amandla iziguli ukuthi zilawule impilo yazo yokuphefumula, kuzivumela ukuthi zihlanganyele emisebenzini yansuku zonke ngokuzethemba nangokukhululeka.

Izwa umehluko nge-Doxofylline - umlingani othembekile ekulweni nezifo zokuphefumula. Xhumana nomhlinzeki wakho wezempilo namuhla ukuze ufunde kabanzi mayelana nokuthi i-Doxofylline ingakusiza kanjani ukuphefumula kalula futhi uphile kangcono.


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