I-H-GLU(OET)-OH (CAS# 1119-33-1)
Sethula i-H-GLU(OET)-OH (I-CAS# 1119-33-1), inhlanganisela esezingeni eliphezulu eyenza izinguquko emkhakheni we-biochemistry kanye nocwaningo lwezemithi. Lo mkhiqizo osuselwe ku-glutamic acid, oklanyelwe ukuthuthukisa ukunyibilika kanye ne-bioavailability yama-ejenti okwelapha. Ngesakhiwo sayo esiyingqayizivele, i-H-GLU(OET)-OH inikeza inkundla eguquguqukayo yokuthuthukiswa kwezidakamizwa, okuyenza ibe ithuluzi elibalulekile kubacwaningi nabakhi bezinto ngokufanayo.
I-H-GLU(OET)-OH ibonakala ngokuzinza kwayo okukhethekile nokuhambisana nezinhlelo ezihlukahlukene zebhayoloji. Ukuguqulwa kwayo kwe-ethyl ester akuthuthukisi nje kuphela ukuncibilika ezindaweni ezinamanzi kodwa futhi kusiza ukufakwa kalula ekwakhiweni okuyinkimbinkimbi. Lokhu kuyenza ibe ikhandidethi elifanele lezicelo ezinhlelweni zokulethwa kwezidakamizwa, lapho ukukhulisa ukusebenza kahle kwezithako ezisebenzayo zemithi kubalulekile.
Ngaphezu kwezinzuzo zayo zokuncibilika, i-H-GLU(OET)-OH ibonisa izakhiwo ezinhle ze-pharmacokinetic, okuvumela ukumuncwa okuthuthukisiwe nokusabalalisa ngaphakathi komzimba. Le nhlanganisela inenzuzo ikakhulukazi ekuthuthukisweni kwezindlela zokwelapha ezisekelwe ku-peptide, lapho ukuthuthukiswa kokulethwa kwama-peptide e-bioactive kungaba nomthelela omkhulu emiphumeleni yokwelapha.
Abacwaningi bazokwazisa ukusetshenziswa kalula nokuphathwa kwe-H-GLU(OET)-OH, njengoba itholakala ngokuhlanzeka okuphezulu futhi ingahlanganiswa ngaphandle komthungo kumaphrothokholi wokuhlola ahlukahlukene. Kungakhathaliseki ukuthi usebenza ekutholakaleni kwezidakamizwa, ekuthuthukisweni kokwakhiwa, noma ocwaningweni lwezemfundo, i-H-GLU(OET)-OH isilungele ukuba yisisekelo elabhorethri yakho.
Vula amandla ocwaningo lwakho nge-H-GLU(OET)-OH (CAS#1119-33-1). Izwa umehluko ongenziwa yile nhlanganisela emisha kumaphrojekthi akho, futhi uthathe igxathu eliya phambili ekufuneni izixazululo zokwelapha ezisebenzayo nezisebenzayo. Yamukela ikusasa le-biochemistry nge-H-GLU(OET)-OH, lapho isayensi ihlangana nokuqamba okusha.